Mutasem O. Taha: шукати на сайті Z-Library

Taha, Mutasem O., AlDamen, Murad A.

Рік:

2013

Мова:

english

Файл:

PDF, 2.80 MB

english, 2013

Effects of Variable Docking Conditions and Scoring Functions on Corresponding Protein-Aligned Comparative Molecular Field Analysis Models Constructed from Diverse Human Protein Tyrosine Phosphatase 1B Inhibitors

Журнал:

Journal of Medicinal Chemistry

Рік:

2005

Мова:

english

Файл:

PDF, 6.24 MB

english, 2005

Tryptophan and thiosemicarbazide derivatives: design, synthesis, and biological evaluation as potential β-d-galactosidase and β-d-glucosidase inhibitors

Abu Khalaf, Reema, Abdula, Ahmed Mutanabbi, Mubarak, Mohammad S., Taha, Mutasem O.

Журнал:

Medicinal Chemistry Research

Рік:

2015

Мова:

english

Файл:

PDF, 4.20 MB

english, 2015

Synthesis of Chitosan Succinate and Chitosan Phthalate and Their Evaluation as Suggested Matrices in Orally Administered, Colon-Specific Drug Delivery Systems

Khaled Aiedeh, Mutasem O. Taha

Журнал:

Archiv der Pharmazie

Рік:

1999

Мова:

english

Файл:

PDF, 96 KB

english, 1999

Discovery of DPP IV Inhibitors by Pharmacophore Modeling and QSAR Analysis followed by in silico Screening

Ihab M. Al-masri, Mohammad K. Mohammad, Mutasem O. Taha

Журнал:

ChemMedChem

Рік:

2008

Мова:

english

Файл:

PDF, 722 KB

english, 2008

Discovery of new β-D-galactosidase inhibitors via pharmacophore modeling and QSAR analysis followed by in silico screening

Ahmed Mutanabbi Abdula, Reema Abu Khalaf, Mohammad S. Mubarak, Mutasem O. Taha

Журнал:

Journal of Computational Chemistry

Рік:

2011

Мова:

english

Файл:

PDF, 1.30 MB

english, 2011

Effect of ionic crosslinking on the drug release properties of chitosan diacetate matrices

Khaled M. Aiedeh, Mutasem O. Taha, Yusuf Al-Hiari, Yasser Bustanji, Hatim S. AlKhatib

Журнал:

Journal of Pharmaceutical Sciences

Рік:

2007

Мова:

english

Файл:

PDF, 135 KB

english, 2007

Synthesis and in vitro behavior of iron-crosslinked N-methyl and N-benzyl hydroxamated derivatives of alginic acid as controlled release carriers

Hatim S. AlKhatib, Mutasem O. Taha, Khaled M. Aiedeh, Yasser Bustanji, Bassam Sweileh

Журнал:

European Polymer Journal

Рік:

2006

Мова:

english

Файл:

PDF, 280 KB

english, 2006

QSPR modeling of pseudoternary microemulsions formulated employing lecithin surfactants: Application of data mining, molecular and statistical modeling

Mutasem O. Taha, Heba Abdel-Halim, Mutasim Al-Ghazawi, Enam Khalil

Журнал:

International Journal of Pharmaceutics

Рік:

2005

Мова:

english

Файл:

PDF, 381 KB

english, 2005

Sodium lauryl sulfate impedes drug release from zinc-crosslinked alginate beads: Switching from enteric coating release into biphasic profiles

Mutasem O. Taha, Wissam Nasser, Adel Ardakani, Hatim S. AlKhatib

Журнал:

International Journal of Pharmaceutics

Рік:

2008

Мова:

english

Файл:

PDF, 858 KB

english, 2008

Discovery of new MurF inhibitors via pharmacophore modeling and QSAR analysis followed by in-silico screening

Mutasem O. Taha, Naji Atallah, Amal G. Al-Bakri, Catherine Paradis-Bleau, Hiba Zalloum, Khaled S. Younis, Roger C. Levesque

Журнал:

Afaf Al-Nadaf, Ghassan Abu Sheikha, Mutasem O. Taha

Рік:

2008

Мова:

english

Файл:

PDF, 1014 KB

english, 2008

Elaborate ligand-based pharmacophore exploration and QSAR analysis guide the synthesis of novel pyridinium-based potent β-secretase inhibitory leads

Журнал:

Maha Habash, Mutasem O. Taha

Рік:

2010

Мова:

english

Файл:

PDF, 1.94 MB

english, 2010

Ligand-based modelling followed by synthetic exploration unveil novel glycogen phosphorylase inhibitory leads

Журнал:

Mutasem O. Taha, Amal G. Al-Bakri, Waleed A. Zalloum

Рік:

2011

Мова:

english

Файл:

PDF, 5.12 MB

english, 2011

Discovery of potent inhibitors of pseudomonal quorum sensing via pharmacophore modeling and in silico screening

Журнал:

Bioorganic & Medicinal Chemistry Letters

Рік:

2006

Мова:

english

Файл:

PDF, 896 KB

english, 2006

Ligand-based assessment of factor Xa binding site flexibility via elaborate pharmacophore exploration and genetic algorithm-based QSAR modeling

Mutasem O. Taha, Amjad M. Qandil, Dhia D. Zaki, Murad A. AlDamen

Журнал:

Areej Abu-Hammad, Waleed A. Zalloum, Hiba Zalloum, Ghassan Abu-Sheikha, Mutasem O. Taha

Рік:

2005

Мова:

english

Файл:

PDF, 2.02 MB

english, 2005

Homology modeling of MCH1 receptor and validation by docking/scoring and protein-aligned CoMFA

Журнал:

Belal O. Al-Najjar, Habibah A. Wahab, Tengku Sifzizul Tengku Muhammad, Alexander Chong Shu-Chien, Nur Adelina Ahmad Noruddin, Mutasem O. Taha

Рік:

2009

Мова:

english

Файл:

PDF, 1.58 MB

english, 2009

Discovery of new nanomolar peroxisome proliferator-activated receptor γ activators via elaborate ligand-based modeling

Журнал:

Mutasem O. Taha, Yasser Bustanji, Amal G. Al-Bakri, Al-Motassem Yousef, Waleed A. Zalloum, Ihab M. Al-Masri, Naji Atallah

Рік:

2011

Мова:

english

Файл:

PDF, 1.35 MB

english, 2011

Discovery of new potent human protein tyrosine phosphatase inhibitors via pharmacophore and QSAR analysis followed by in silico screening

Журнал:

Areej M. Abu Hammad, Fatma U. Afifi, Mutasem O. Taha

Рік:

2007

Мова:

english

Файл:

PDF, 2.19 MB

english, 2007

Combining docking, scoring and molecular field analyses to probe influenza neuraminidase–ligand interactions

Журнал:

Hiba M. Zalloum, Mutasem O. Taha

Рік:

2007

Мова:

english

Файл:

PDF, 2.34 MB

english, 2007

Development of predictive in silico model for cyclosporine- and aureobasidin-based P-glycoprotein inhibitors employing receptor surface analysis

Журнал:

Afaf H. Al-Nadaf, Mutasem O. Taha

Рік:

2008

Мова:

english

Файл:

PDF, 1.41 MB

english, 2008

Discovery of new renin inhibitory leads via sequential pharmacophore modeling, QSAR analysis, in silico screening and in vitro evaluation

Журнал:

Harry Heaney*, Mutasem O Taha, Alexandra M.Z Slawin

Рік:

2011

Мова:

english

Файл:

PDF, 1.26 MB

english, 2011

The Oxidation of Homophthalimide Derivatives by Dioxygen in Alkaline Media and Cleavage-Cyclisation Reactions

Журнал:

Tetrahedron Letters

Рік:

1997

Мова:

english

Файл:

PDF, 627 KB

english, 1997

The bis(homoallylic) stabilisation of an acyliminium ion and reactions with nucleophiles

Harry Heaney, Mutasem O. Taha

Журнал:

Tetrahedron Letters

Рік:

1998

Мова:

english

Файл:

PDF, 280 KB

english, 1998

Discovery of new β-d-glucosidase inhibitors via pharmacophore modeling and QSAR analysis followed by in silico screening

Reema Abu Khalaf, Ahmed Mutanabbi Abdula, Mohammad S. Mubarak, Mutasem O. Taha

Журнал:

Journal of Molecular Modeling

Рік:

2011

Мова:

english

Файл:

PDF, 1.52 MB

english, 2011

Elaborate ligand-based modeling reveal new submicromolar Rho kinase inhibitors

Rand Shahin, Saja AlQtaishat, Mutasem O. Taha

Журнал:

Journal of Computer-Aided Molecular Design

Рік:

2012

Мова:

english

Файл:

PDF, 1.08 MB

english, 2012

Discovery of new cholesteryl ester transfer protein inhibitors via ligand-based pharmacophore modeling and QSAR analysis followed by synthetic exploration

Reema Abu Khalaf, Ghassan Abu Sheikha, Yasser Bustanji, Mutasem O. Taha

Журнал:

Mahmoud A. Al-Sha’er, Mutasem O. Taha

Рік:

2010

Мова:

english

Файл:

PDF, 1.35 MB

english, 2010

Discovery of novel CDK1 inhibitors by combining pharmacophore modeling, QSAR analysis and in silico screening followed by in vitro bioassay

Журнал:

Mutasem O. Taha, Mai Tarairah, Hiba Zalloum, Ghassan Abu-Sheikha

Рік:

2010

Мова:

english

Файл:

PDF, 1.57 MB

english, 2010

Pharmacophore and QSAR modeling of estrogen receptor β ligands and subsequent validation and in silico search for new hits

Журнал:

Harry Heaney, Mutasem O Taha

Рік:

2010

Мова:

english

Файл:

PDF, 966 KB

english, 2010

N-Acyliminium ion cyclisation versus rearrangement. The synthesis of 13,13-dimethylberberines and 3,4-dimethylisoquinolin-1-ones

Журнал:

Tetrahedron Letters

Рік:

2000

Мова:

english

Файл:

PDF, 119 KB

english, 2000

In Silico Screening for Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors Using Physicochemical Filters and High-Throughput Docking Followed by In Vitro Evaluation

Yasser Bustanji, Ihab M. Al-Masri, Ahmad Qasem, Amal G. Al-Bakri, Mutasem Omar Taha

Журнал:

Chemical Biology & Drug Design

Рік:

2009

Мова:

english

Файл:

PDF, 308 KB

english, 2009

Ethosuximide and Phenobarbital Promote Wound Healing via Enhancing Collagenization

Dema M. Ajwee, Ahmad M. Disi, Eyad A. Qunaibi, Mutasem O. Taha

Журнал:

Chemical Biology & Drug Design

Рік:

2012

Мова:

english

Файл:

PDF, 454 KB

english, 2012

Discovery of New Antifungal Leads via Pharmacophore Modeling and QSAR Analysis of Fungal N-Myristoyl Transferase Inhibitors Followed by In Silico Screening

Mutasem O. Taha, Amjad M. Qandil, Tariq Al-Haraznah, Reema Abu Khalaf, Hiba Zalloum, Amal G. Al-Bakri

Журнал:

Chemical Biology & Drug Design

Рік:

2011

Мова:

english

Файл:

PDF, 1.11 MB

english, 2011

Docking-Based Comparative Intermolecular Contacts Analysis as New 3-D QSAR Concept for Validating Docking Studies and in Silico Screening: NMT and GP Inhibitors as Case Studies

Taha, Mutasem O., Habash, Maha, Al-Hadidi, Zeina, Al-Bakri, Amal, Younis, Khaled, Sisan, Suhaib

Журнал:

Journal of Chemical Information and Modeling

Рік:

2011

Мова:

english

Файл:

PDF, 1.47 MB

english, 2011

Rational exploration of new pyridinium-based HSP90α inhibitors tailored to thiamine structure

Mahmoud A. Al-Sha’er, Mutasem O. Taha

Журнал:

Medicinal Chemistry Research

Рік:

2012

Мова:

english

Файл:

PDF, 881 KB

english, 2012

Elaborate ligand-based modeling and subsequent synthetic exploration unveil new nanomolar Ca2+/calmodulin-dependent protein kinase II inhibitory leads

Rand Shahin, Mutasem O. Taha

Журнал:

Mohammad K. Mohammad, Ihab M. Al-masri, Mutasem O. Taha, Mohamed A.S. Al-Ghussein, Hatim S. AlKhatib, Samer Najjar, Yasser Bustanji

Рік:

2012

Мова:

english

Файл:

PDF, 3.27 MB

english, 2012

Olanzapine inhibits glycogen synthase kinase-3β: An investigation by docking simulation and experimental validation

Журнал:

European Journal of Pharmacology

Рік:

2008

Мова:

english

Файл:

PDF, 418 KB

english, 2008

Metal ion / Pyridinedicarboxylate Polymer composites as inhibitors of bacterial biofilm formation: Category: Scientific free paper

Suhair Saleh, Bassam Sweileh, Sami Taha, Mutasem Taha

Журнал:

Journal of Infection

Рік:

2011

Мова:

english

Файл:

PDF, 43 KB

english, 2011

Extensive ligand-based modeling and in silico screening reveal nanomolar inducible nitric oxide synthase (iNOS) inhibitors

Ghadeer A.R.Y. Suaifan, Mayyada Shehadehh, Hebah Al-Ijel, Mutasem O. Taha

Журнал:

Khaled Aiedeh, Mutasem O. Taha

Рік:

2012

Мова:

english

Файл:

PDF, 6.97 MB

english, 2012

Synthesis of iron-crosslinked chitosan succinate and iron-crosslinked hydroxamated chitosan succinate and their in vitro evaluation as potential matrix materials for oral theophylline sustained-release beads

Журнал:

European Journal of Pharmaceutical Sciences

Рік:

2001

Мова:

english

Файл:

PDF, 404 KB

english, 2001

Development of quantitative structure–property relationship models for pseudoternary microemulsions formulated with nonionic surfactants and cosurfactants: application of data mining and molecular modeling

Mutasem O. Taha, Mutasim Al-Ghazawi, Hend Abu-Amara, Enam Khalil

Журнал:

European Journal of Pharmaceutical Sciences

Рік:

2002

Мова:

english

Файл:

PDF, 452 KB

english, 2002

Synthesis and biological activity assays of some new N1-(flavon-7-yl)amidrazone derivatives and related congeners

Abu-Aisheh, Marwa N., Mustafa, Mohammad S., El-Abadelah, Mustafa M., Naffa, Randa G., Ismail, Said I., Zihlif, Malek A., Taha, Mutasem O., Mubarak, Mohammad S.

Журнал: